Caffeine is a central nervous system stimulant that temporarily wards off drowsiness and boosts alertness and energy.

Ephedra Extract is extracted from the plant Ephedra sinica, It has been used in traditional Chinese medicine for the treatment of asthma and hay fever. Ephedra is used both as a stimulant and a thermogenic, which stimulates the brain, increases heart rate, increases blood pressure and expands bronchial tubes (making breathing easier). These effects are due to its ephedrine and pseudoephedrine content. Research also shows that it can be used as a precursor in the illicit manufacture of methamphetamine. Ephedra extracts are also used by athletes to enhance athletic performance. It is also used in supplements for weight loss.

Glucuronolactone is also used as a detoxicant but is actually a natural chemical produced by glucose metabolism in the human liver.

Nettle has tonic, anti-inflammatory, hemostatic, and diuretic properties. Nettle has been used to treat rheumatism, eczema, arthritis, gout, and anemia. Nettle is very effective in treating urinary tract infections. An infusion of the nettle leaves can be used for inflammatory diseases of the lower urinary tract and also is effective for treating certain individuals with allergic reactions to hay fever.It helps the body to eliminate waste products and prevents fluid retention. Nettle's properties have been beneficial for coughs and have been used to get rid of phlegm from the lungs and stomach. Nettle helps draw body tissues together and control bleeding. Nettle leaf is used in a simple infusion as a tonic decoction to cleanse the blood. Nettle is also used as a specific for treating cases of childhood eczema; it's especially useful for nervous eczema. Nettle leaves contain iron and vitamin C and is sometimes used for treating anemia and poor circulation.

Phenylethlamine HCL is a salt of phenylethylamine. It is a crystalline solid and is formed by treating phenylethylamine with HCl. Its IUPAC name is 2 phenylethylamine HCl. The scientific name elucidates its chemical structure. It is an aromatic compound meaning that it has a basic benzene ring. It further has a two carbon chain attached at position 2 of the ring and the chain terminates in an amino group. It occurs naturally in some foods like chocolates but the food item might get metabolized too quickly sometimes for it to have a significant effect on the body. This substance has quite profound effects on the level of dopamine in the central nervous system, provided it passes the blood brain barrier. It increases dopamine level and at the same time inhibits dopamine transmitters resulting in a buildup of dopamine in the brain. While excessive levels of dopamine in the CNS are not healthy, the neurotransmitter does regulate cognition, mood, voluntary movement and other brain functions.

Picamilon , also known as nicotinoyl-GABAm Pycamilon, Pikamilon, is formed by combining niacin with GABA. It is basically a dietary supplement. All-Union Scientific Research Institute of the Soviet Union developed this dietary supplement in 1969. It was further studied in Japan and Russia as a prodrug of GABA. In the United States, picamilon is sold as a dietary supplement whereas in Russia, the same drug picamilon is sold as a prescription drug. Picamilon hydrolyzes into GABA and niacin by crossing the blood brain barrier. In theory, the released GABA receptors would activate and potentially produce an anxiolytic response. It also releases a second component known as niacin. Niacin then acts as a strong vasodilator. This niacin then comes in use for the treatment of migraine heaaches.

Synephrine is an active compound that may be found in the fruit called Citrus aurantium or Zhi Shi in Chinese. Its chemical composition is similar to ephedrine and pseudo-ephedrine that may be found in most over the counter cold or allergy medications, weight loss and energy supplements. Unlike ephedrine, Synephrine is considered to be semi-selective sympathomimetic that targets tissues such as fats instead of the heart. It also helps the metabolism without the negative effects of ephedrine to the nervous system. It also increases the energy level, helps the body burn fat and promotes weight loss. It also aids the body to increase the quickness of caloric expenditure.

Xanthinol Nicotinate, a very potent form of niacin.

Yohimbine HCL, sometimes called yohimbine hydrochloride, yohimbe, or yohimbe bark, is an herbal supplement which serves as a stimulant and possible aphrodisiac for users. Yohimbine has also been shown to be successful in treating erectile dysfunction and impotence in men. It may serve to boost the sex drive of those who take it for aphrodisiac purposes. Some people are recommended to take yohimbine to combat their lower sex drives caused by antidepressants. Yohimbine has also been shown to help blood pressure levels and assist in weight loss. For these reasons, yohimbine is a popular supplement amongst athletes as well as many others wishing to improve their health.